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Ly-215,840

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Title: Ly-215,840  
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Subject: 5-HT7 receptor, Eli Lilly and Company, RS-56812, BRL-54443, MPPF
Collection: 5-Ht2 Antagonists, Eli Lilly and Company, Ergolines
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Ly-215,840

LY-215,840
Systematic (IUPAC) name
(6aR,9R,10aR)-N-((1S,2R)-2-hydroxycyclopentyl)-4-isopropyl-7-methyl-4,6,6a,7,8,9,10,10a-octahydroindolo[4,3-fg]quinoline-9-carboxamide
Identifiers
CAS Registry Number
PubChem CID:
IUPHAR/BPS
Chemical data
Formula C24H33N3O2
Molecular mass 395.54 g/mol

LY-215,840 is an ergoline derivative drug developed by Eli Lilly, which acts as a potent and selective antagonist at the serotonin 5-HT2 and 5-HT7 receptors. It has anti-hypertensive and muscle relaxant effects in animal studies.[1][2][3][4][5][6][7][8]


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